联硼酸频那醇酯合成路线

参考文献

Xuanzhu Pharma Co., Ltd.; WU, Frank; ZHANG, Yan
Patent: EP2719697 A1, 2014 ;
Location in patent: Paragraph 0176; 0179; 0180 ;

1162262-35-2

参考文献

AMGEN INC.; DRANSFIELD, Paul, John; GONZALEZ LOPEZ DE TURISO, Felix; KOHN, Todd, J.; PATTAROPONG, Vatee; SIMARD, Jillian, L.
Patent: WO2012/3283 A1, 2012 ;
Location in patent: Page/Page column 228-229 ;
WO 2012/003283 A1

709652-82-42-氨基-5-溴-3-腈基吡啶+

73183-34-3联硼酸频那醇酯

1246372-66-62-氨基-5-(4,4,5,5-四甲基-1,3,2-二噁硼烷-2-基)吡啶-3-甲腈

参考文献

OTSUKA PHARMACEUTICAL CO., LTD.; ABUDUSAIMI, Mamuti; YE, Fangguo; SUN, Jiangqin; MIYAMOTO, Hisashi; CHENG, Jay-Fei; OKA, Daisuke
Patent: WO2013/29548 A1, 2013 ;
Location in patent: Page/Page column 87 ;

5910-12-33-溴吡唑并[1,5-a]吡啶+

73183-34-3联硼酸频那醇酯

1207557-48-93-(4,4,5,5-四甲基-1,3,2-二噁硼烷-2-基)h-吡唑并[1,5-a]吡啶

参考文献

ALMIRALL, S.A.; BACH TANA, Jordi; PAGES SANTACANA, Lluis, Miquel; TALTAVULL MOLL, Joan; EASTWOOD, Paul, Robert; GONZALEZ RODRIGUES, Jacob; GIULIO MATASSA, Victor
Patent: WO2011/101161 A1, 2011 ;
Location in patent: Page/Page column 103 ;
WO 2011/101161 A1

1435-43-43,5-二氟氯苯+

73183-34-3联硼酸频那醇酯

1165935-84-1

参考文献

Robbins, Daniel W.; Hartwig, John F.
Organic Letters, 2012 , vol. 14, # 16 p. 4266 - 4269

1174038-64-2+

73183-34-3联硼酸频那醇酯

1174038-65-31-(苯基磺酰基)-3-(4,4,5,5-四甲基-1,3,2-二噁硼烷-2-基)-1H-吡咯并[2,3-c]吡啶

参考文献

Merck Patent Gesellschaft Mit Beschrankter Haftung
Patent: US2010/292262 A1, 2010 ;
Location in patent: Page/Page column 13-14 ;

404827-77-63-氨基-6-溴-1H-吲唑+

73183-34-3联硼酸频那醇酯

1187968-75-76-(4,4,5,5-四甲基-1,3,2-二氧杂环己硼烷-2-基)-3-氨基-1H-吲唑

参考文献

Deng, Xianming; Zhou, Wenjun; Weisberg, Ellen; Wang, Jinhua; Zhang, Jianming; Sasaki, Takaaki; Nelson, Erik; Griffin, James D.; Jaenne, Pasi A.; Gray, Nathanael S.
Bioorganic and Medicinal Chemistry Letters, 2012 , vol. 22, # 14 p. 4579 - 4584

928775-04-6+

73183-34-3联硼酸频那醇酯

1201644-51-0

参考文献

Gordeev, Mikhail Fedorovich; Yuan, Zhengyu; Liu, Jinqian; Wang, Qiang
Patent: US2010/69441 A1, 2010 ;
Location in patent: Page/Page column 36-37 ;

1227177-83-4+

73183-34-3联硼酸频那醇酯

1227068-67-8

参考文献

AMGEN INC.
Patent: US2010/160280 A1, 2010 ;
Location in patent: Page/Page column 161 ;

214342-63-9+

73183-34-3联硼酸频那醇酯

1160790-84-0

参考文献

PROLYSIS LTD
Patent: WO2009/74812 A1, 2009 ;
Location in patent: Page/Page column 73 ;
WO 2009/074812 A1