联硼酸频那醇酯合成路线

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ASTRAZENECA AB; ASTEX THERAPEUTICS LTD
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150-19-63-甲氧基苯酚+

73183-34-3联硼酸频那醇酯

906008-22-83-甲氧基-5-(4,4,5,5-四甲基-1,3,2-二噁硼烷-2-基)苯酚

参考文献

Ishikawa, Shunpei; Manabe, Kei
Chemical Communications, 2006 , # 24 p. 2589 - 2591

4532-25-67-氯咪唑并[1,2-a]吡啶+

73183-34-3联硼酸频那醇酯

908268-52-0咪唑并[1,2-a]吡啶-7-硼酸频那醇酯

参考文献

Aicher, Thomas Daniel; Anzeveno, Peter Biagio; Li, Renhua; Krasutsky, Alexei Pavlovych; Mabry, Thomas Edward; Saeed, Ashraf; Snyder, Nancy June; Stephenson, Gregory Alan; Tian, Hongqi; Wallace, Owen Brendan; Winneroski, JR., Leonard Larry; Xu, Yanping
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808744-34-57-溴咪唑并[1,2-a]吡啶+

73183-34-3联硼酸频那醇酯

908268-52-0咪唑并[1,2-a]吡啶-7-硼酸频那醇酯

参考文献

GLAXOSMITHKLINE LLC; ADAMS, Nicholas, David; CHAUDHARI, Amita, M.; KIESOW, Terence, John; McSHERRY, Allison, K.; MOORE, Michael, Lee; PARRISH, Cynthia, Ann; REIF, Alexander, Joseph; RIDGERS, Lance, Howard
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55289-35-52-溴-6-硝基甲苯+

73183-34-3联硼酸频那醇酯

910235-64-22-甲基-3-硝基苯硼酸频那醇酯

参考文献

F. HOFFMANN-LA ROCHE AG
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73183-34-3联硼酸频那醇酯+

673485-54-65-溴-N,N-二乙基吡啶甲酰胺

911227-46-86-二乙基氨基甲酰吡啶-3-硼酸频那醇酯

参考文献

Bourdonnec, Bertrand Le; Windh, Rolf T.; Leister, Lara K.; Zhou, Q. Jean; Ajello, Christopher W.; Gu, Minghua; Chu, Guo-Hua; Tuthill, Paul A.; Barker, William M.; Koblish, Michael; Wiant, Daniel D.; Graczyk, Thomas M.; Belanger, Serge; Cassel, Joel A.; Feschenko, Marina S.; Brogdon, Bernice L.; Smith, Steven A.; Derelanko, Michael J.; Kutz, Steve; Little, Patrick J.; Dehaven, Robert N.; DeHaven-Hudkins, Diane L.; Dolle, Roland E.
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7606-13-5+

73183-34-3联硼酸频那醇酯

911227-46-86-二乙基氨基甲酰吡啶-3-硼酸频那醇酯

参考文献

Hurst, Timothy E.; Macklin, Todd K.; Becker, Maike; Hartmann, Eduard; Kuegel, Wolfgang; Parisienne-LaSalle, Jean-Christophe; Batsanov, Andrei S.; Marder, Todd B.; Snieckus, Victor
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911227-44-6+

73183-34-3联硼酸频那醇酯

911228-63-2

参考文献

Bourdonnec, Bertrand Le; Windh, Rolf T.; Leister, Lara K.; Zhou, Q. Jean; Ajello, Christopher W.; Gu, Minghua; Chu, Guo-Hua; Tuthill, Paul A.; Barker, William M.; Koblish, Michael; Wiant, Daniel D.; Graczyk, Thomas M.; Belanger, Serge; Cassel, Joel A.; Feschenko, Marina S.; Brogdon, Bernice L.; Smith, Steven A.; Derelanko, Michael J.; Kutz, Steve; Little, Patrick J.; Dehaven, Robert N.; DeHaven-Hudkins, Diane L.; Dolle, Roland E.
Journal of Medicinal Chemistry, 2009 , vol. 52, # 18 p. 5685 - 5702

387-44-07-氟吲哚+

73183-34-3联硼酸频那醇酯

912331-75-0

参考文献

ELI LILLY AND COMPANY
Patent: WO2006/107784 A1, 2006 ;
Location in patent: Page/Page column 66 ;
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882670-77-1+

73183-34-3联硼酸频那醇酯

913067-91-1

参考文献

DiMauro, Erin F.; Newcomb, John; Nunes, Joseph J.; Bemis, Jean E.; Boucher, Christina; Buchanan, John L.; Buckner, William H.; Cee, Victor J.; Chai, Lilly; Deak, Holly L.; Epstein, Linda F.; Faust, Ted; Gallant, Paul; Geuns-Meyer, Stephanie D.; Gore, Anu; Gu, Yan; Henkle, Brad; Hodous, Brian L.; Hsieh, Faye; Huang, Xin; Kim, Joseph L.; Lee, Josie H.; Martin, Matthew W.; Masse, Craig E.; McGowan, David C.; Metz, Daniela; Mohn, Deanna; Morgenstern, Kurt A.; Oliveira-Dos-Santos, Antonio; Patel, Vinod F.; Powers, David; Rose, Paul E.; Schneider, Stephen; Tomlinson, Susan A.; Tudor, Yan-Yan; Turci, Susan M.; Welcher, Andrew A.; White, Ryan D.; Zhao, Huilin; Zhu, Li; Zhu, Xiaotian
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