联硼酸频那醇酯合成路线

参考文献

Malo-Forest, Bianca; Landelle, Gregory; Roy, Jessye-Ann; Lacroix, Jacques; Gaudreault, Rene C.; Paquin, Jean-Francois
Bioorganic and Medicinal Chemistry Letters, 2013 , vol. 23, # 6 p. 1712 - 1715

73183-34-3联硼酸频那醇酯+

179898-34-13-溴-5-氟苯腈

935685-88-43-氟-5-(4,4,5,5-四甲基-1,3,2-二噁硼烷-2-基)苯甲腈

参考文献

AiCuris GmbH and Co. KG; Thede, Kai; Greschat, Susanne; Gericke, Kersten Matthias; Wildum, Steffen; Paulsen, Daniela
Patent: US2013/45999 A1, 2013 ;
Location in patent: Paragraph 0224; 0225; 0226; 0227 ;

936923-58-95-溴-1,2-苯并异噻唑-3-羧酸乙酯+

73183-34-3联硼酸频那醇酯

936923-42-15-(4,4,5,5-四甲基-1,3,2-二氧硼烷)-1,2-苯并异噻唑-3-羧酸乙酯

参考文献

MEMORY PHARMACEUTICALS CORPORATION
Patent: WO2007/56582 A1, 2007 ;
Location in patent: Page/Page column 70 ;
WO 2007/056582 A1

73183-34-3联硼酸频那醇酯

937366-54-6吲哚-5-硼酸频那醇酯

参考文献

Takagi, Jun; Sato, Kazuaki; Hartwig, John F; Ishiyama, Tatsuo; Miyaura, Norio
Tetrahedron Letters, 2002 , vol. 43, # 32 p. 5649 - 5651

937591-28-11-(7-溴-3,4-二氢异喹啉-2(1h)-基)乙酮+

73183-34-3联硼酸频那醇酯

937591-29-2

参考文献

ASTRAZENECA AB; ASTEX THERAPEUTICS LTD
Patent: WO2007/58602 A2, 2007 ;
Location in patent: Page/Page column 77-78 ;
WO 2007/058602 A2

73183-34-3联硼酸频那醇酯+

937591-81-6

937591-82-7

参考文献

ASTRAZENECA AB; ASTEX THERAPEUTICS LTD
Patent: WO2007/58602 A2, 2007 ;
Location in patent: Page/Page column 112-113 ;
WO 2007/058602 A2

3722-78-9+

73183-34-3联硼酸频那醇酯

937591-99-6

参考文献

ASTRAZENECA AB; ASTEX THERAPEUTICS LTD
Patent: WO2007/73284 A1, 2007 ;
Location in patent: Page/Page column 46 ;
WO 2007/073284 A1

98612-93-21-(4-溴苯甲酰基)哌啶+

73183-34-3联硼酸频那醇酯

938043-31-3

参考文献

Patel, Gautam; Karver, Caitlin E.; Behera, Ranjan; Guyett, Paul J.; Sullenberger, Catherine; Edwards, Peter; Roncal, Norma E.; Mensa-Wilmot, Kojo; Pollastri, Michael P.
Journal of Medicinal Chemistry, 2013 , vol. 56, # 10 p. 3820 - 3832

321-23-32-氟-4-溴硝基苯+

73183-34-3联硼酸频那醇酯

939968-60-23-氟-4-硝基苯硼酸频那醇酯

参考文献

ABBOTT LABORATORIES
Patent: WO2008/63287 A2, 2008 ;
Location in patent: Page/Page column 54 ;

2369-13-33-氟-4-硝基苯胺+

73183-34-3联硼酸频那醇酯

939968-60-23-氟-4-硝基苯硼酸频那醇酯

参考文献

Qiu, Di; Wang, Shuai; Tang, Shengbo; Meng, He; Jin, Liang; Mo, Fanyang; Zhang, Yan; Wang, Jianbo
Journal of Organic Chemistry, 2014 , vol. 79, # 5 p. 1979 - 1988