联硼酸频那醇酯合成路线

943324-08-12-甲基-1-苯磺酰基-3-(4,4,5,5-四甲基-1,3,2-二噁硼烷-2-基)-1H-吡咯并[2,3-B]吡啶

参考文献

SMITHKLINE BEECHAM CORPORATION
Patent: WO2007/76423 A2, 2007 ;
Location in patent: Page/Page column 171 ;
WO 2007/076423 A2

560082-53-36-溴-8-氟-2H-苯并[b][1,4]恶嗪-3(4H)-酮+

73183-34-3联硼酸频那醇酯

943994-40-9

参考文献

Hasui, Tomoaki; Ohra, Taiichi; Ohyabu, Norio; Asano, Kouhei; Matsui, Hideki; Mizukami, Atsushi; Habuka, Noriyuki; Sogabe, Satoshi; Endo, Satoshi; Siedem, Christopher S.; Tang, Tony P.; Gauthier, Cassandra; De Meese, Lisa A.; Boyd, Steven A.; Fukumoto, Shoji
Bioorganic and Medicinal Chemistry, 2013 , vol. 21, # 19 p. 5983 - 5994

121564-97-46-溴-8-甲基-4H-1,4-苯并恶嗪-3-酮+

73183-34-3联硼酸频那醇酯

943994-87-4

参考文献

TAKEDA PHARMACEUTICAL COMPANY LIMITED
Patent: WO2007/77961 A2, 2007 ;
Location in patent: Page/Page column 361 ;
WO 2007/077961 A2

124840-58-0甲基(3-碘-4-甲氧基苯基)乙酸酯+

73183-34-3联硼酸频那醇酯

944317-65-12-(4-甲氧基-3-(4,4,5,5-四甲基-1,3,2-二噁硼烷-2-基)苯基)乙酸甲酯

参考文献

CHONG KUN DANG PHARMACEUTICAL CORP.; LEE, Seohee; OH, Jungtaek; LEE, Jaekwang; LEE, Jaewon; BAE, Suyeal; HA, Nina; LEE, Sera
Patent: WO2012/141487 A2, 2012 ;
Location in patent: Page/Page column 34; 74 ;
WO 2012/141487 A2

19626-36-9+

73183-34-3联硼酸频那醇酯

944317-65-12-(4-甲氧基-3-(4,4,5,5-四甲基-1,3,2-二噁硼烷-2-基)苯基)乙酸甲酯

参考文献

Ghosh, Samir; Kumar, A. Sanjeev; Mehta; Soundararajan
Synthesis, 2009 , # 19 p. 3322 - 3326

885681-61-8+

73183-34-3联硼酸频那醇酯

944317-66-22-氟-5-(甲氧基羰基甲基)苯硼酸频那醇酯

参考文献

AMIRA PHARMACEUTICALS, INC.; HUTCHINSON, John, Howard; SEIDERS, Thomas, Jon; ARRUDA, Jeannie, M.; ROPPE, Jeffrey, Roger
Patent: WO2010/42652 A2, 2010 ;
Location in patent: Page/Page column 102 ;
WO 2010/042652 A2

51839-15-75-碘间苯二甲酸二甲酯+

73183-34-3联硼酸频那醇酯

944392-68-13,5-二甲氧羰基苯硼酸频哪醇酯

参考文献

Park, Jinhee; Wang, Zhiyong U.; Sun, Lin-Bing; Chen, Ying-Pin; Zhou, Hong-Cai
Journal of the American Chemical Society, 2012 , vol. 134, # 49 p. 20110 - 20116

20330-90-95-氯异邻苯二甲酸二甲酯+

73183-34-3联硼酸频那醇酯

944392-68-13,5-二甲氧羰基苯硼酸频哪醇酯

参考文献

Tang, Wenjun; Keshipeddy, Santosh; Zhang, Yongda; Wei, Xudong; Savoie, Jolaine; Patel, Nitinchandra D.; Yee, Nathan K.; Senanayake, Chris H.
Organic Letters, 2011 , vol. 13, # 6 p. 1366 - 1369

51760-21-55-溴异肽酸二甲基酯+

73183-34-3联硼酸频那醇酯

944392-68-13,5-二甲氧羰基苯硼酸频哪醇酯

参考文献

Peng, Yang; Krungleviciute, Vaiva; Eryazici, Ibrahim; Hupp, Joseph T.; Farha, Omar K.; Yildirim, Taner
Journal of the American Chemical Society, 2013 , vol. 135, # 32 p. 11887 - 11894

99-27-45-氨基间苯二甲酸二甲酯+

73183-34-3联硼酸频那醇酯

944392-68-13,5-二甲氧羰基苯硼酸频哪醇酯

参考文献

Qiu, Di; Jin, Liang; Zheng, Zhitong; Meng, He; Mo, Fanyang; Wang, Xi; Zhang, Yan; Wang, Jianbo
Journal of Organic Chemistry, 2013 , vol. 78, # 5 p. 1923 - 1933