联硼酸频那醇酯合成路线

参考文献

Lu, Jie; Guan, Zhong-Zhi; Gao, Jian-Wu; Zhang, Zhan-Hui
Applied Organometallic Chemistry, 2011 , vol. 25, # 7 p. 537 - 541

626-01-73-碘苯胺+

73183-34-3联硼酸频那醇酯

408492-28-43-碘苯硼酸频哪酯

参考文献

Qiu, Di; Jin, Liang; Zheng, Zhitong; Meng, He; Mo, Fanyang; Wang, Xi; Zhang, Yan; Wang, Jianbo
Journal of Organic Chemistry, 2013 , vol. 78, # 5 p. 1923 - 1933

580-17-63-氨基喹啉+

73183-34-3联硼酸频那醇酯

171364-85-53-喹啉硼酸频哪醇酯

参考文献

Qiu, Di; Jin, Liang; Zheng, Zhitong; Meng, He; Mo, Fanyang; Wang, Xi; Zhang, Yan; Wang, Jianbo
Journal of Organic Chemistry, 2013 , vol. 78, # 5 p. 1923 - 1933

91-22-5喹啉+

73183-34-3联硼酸频那醇酯

171364-85-53-喹啉硼酸频哪醇酯

参考文献

Takagi, Jun; Sato, Kazuaki; Hartwig, John F; Ishiyama, Tatsuo; Miyaura, Norio
Tetrahedron Letters, 2002 , vol. 43, # 32 p. 5649 - 5651

20986-40-75-溴烟酸乙酯+

73183-34-3联硼酸频那醇酯

916326-10-83-(乙氧基甲酰基)吡啶-5-硼酸频哪醇酯

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ELI LILLY AND COMPANY
Patent: US2012/184577 A1, 2012 ;
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20986-40-75-溴烟酸乙酯+

73183-34-3联硼酸频那醇酯

916326-10-83-(乙氧基甲酰基)吡啶-5-硼酸频哪醇酯

参考文献

Leblanc, Yves; Cerat, Pascal
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17321-93-62-氨基-5-溴-4-甲基嘧啶+

73183-34-3联硼酸频那醇酯

944401-55-22-氨基-4-甲基嘧啶-5-硼酸频哪酯

参考文献

Genentech, Inc.; Heald, Robert Andrew; McLean, Neville James
Patent: US2014/65136 A1, 2014 ;
Location in patent: Paragraph 0198; 0199 ;

17321-93-62-氨基-5-溴-4-甲基嘧啶+

73183-34-3联硼酸频那醇酯

108-52-12-氨基-4-甲基嘧啶+

944401-55-22-氨基-4-甲基嘧啶-5-硼酸频哪酯

参考文献

Burger, Matthew T.; Pecchi, Sabina; Wagman, Allan; Ni, Zhi-Jie; Knapp, Mark; Hendrickson, Thomas; Atallah, Gordana; Pfister, Keith; Zhang, Yanchen; Bartulis, Sarah; Frazier, Kelly; Ng, Simon; Smith, Aaron; Verhagen, Joelle; Haznedar, Joshua; Huh, Kay; Iwanowicz, Ed; Xin, Xiaohua; Menezes, Daniel; Merritt, Hanne; Lee, Isabelle; Wiesmann, Marion; Kaufman, Susan; Crawford, Kenneth; Chin, Michael; Bussiere, Dirksen; Shoemaker, Kevin; Zaror, Isabel; Maira, Sauveur-Michel; Voliva, Charles F.
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56686-16-95-溴-2,4-二甲氧基嘧啶+

73183-34-3联硼酸频那醇酯

936250-17-8

参考文献

de Vicente Fidalgo, Javier; Li, Jim; Schoenfeld, Ryan Craig; Talamas, Francisco Xavier; Taygerly, Joshua Paul Gergely
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Location in patent: Page/Page column 49-50 ;

24036-52-06-溴-2H-1,4-苯并噁嗪-3(4H)-酮+

73183-34-3联硼酸频那醇酯

943994-02-3

参考文献

WO2010/116282 A1, ;

Page/Page column 55-56 ;
WO 2010/116282 A1