联硼酸频那醇酯合成路线

参考文献

Robbins, Daniel W.; Hartwig, John F.
Angewandte Chemie - International Edition, 2013 , vol. 52, # 3 p. 933 - 937
Angew. Chem., 2012 , vol. 125, # 3 p. 967 - 971,5

83-34-13-甲基吲哚+

73183-34-3联硼酸频那醇酯+

25015-63-8频哪醇硼烷

1072812-35-1

参考文献

Robbins, Daniel W.; Boebel, Timothy A.; Hartwig, John F.
Journal of the American Chemical Society, 2010 , vol. 132, # 12 p. 4068 - 4069

897016-95-4(4-溴-3-氟-苯基)-吗啉-4-基-甲酮+

73183-34-3联硼酸频那醇酯

1092500-69-02-氟-4-(吗啉-4-甲酰基)苯硼酸

参考文献

WO2008/148867 A2, ;

Page/Page column 28-29 ;
WO 2008/148867 A2

53484-15-45-溴-1-甲基-1H-苯并[d]咪唑+

73183-34-3联硼酸频那醇酯

1107627-02-01-甲基-5-(4,4,5,5-四甲基-1,3,2-二硼戊环-2-基)-1H-苯并[d]咪唑

参考文献

TAKEDA PHARMACEUTICAL COMPANY LIMITED; LAWSON, John David; SABAT, Mark; SMITH, Christopher; WANG, Haixia; CHEN, Young K.; KANOUNI, Toufike
Patent: WO2013/148603 A1, 2013 ;
Location in patent: Paragraph 0219-0220 ;

73183-34-3联硼酸频那醇酯

1075249-37-4

参考文献

IRM LLC
Patent: WO2008/134300 A1, 2008 ;
Location in patent: Page/Page column 31-32 ;
WO 2008/134300 A1

2973-80-02-溴-5-羟基苯甲醛+

73183-34-3联硼酸频那醇酯

1038827-60-9

参考文献

ASTRAZENECA AB; ASTRAZENECA UK LIMITED
Patent: WO2008/84223 A2, 2008 ;
Location in patent: Page/Page column 144-145 ;
WO 2008/084223 A2

164513-39-72-甲氧基-4-甲基-5-溴吡啶+

73183-34-3联硼酸频那醇酯

1093951-66-62-甲氧基-4-甲基-5-(4,4,5,5-四甲基-[1,3,2]二噁硼烷-2-基)-吡啶

参考文献

US2008/318943 A1, ;

Page/Page column 73; 75 ;
US 20080318943 A1

88139-91-75-溴-2-羟甲基吡啶+

73183-34-3联硼酸频那醇酯

1078575-71-9

参考文献

Xuanzhu Pharma Co., Ltd.; WU, Frank; ZHANG, Yan
Patent: EP2719697 A1, 2014 ;
Location in patent: Paragraph 0164-0166 ;

5053-43-02-甲基嘧啶+

73183-34-3联硼酸频那醇酯

1052686-67-5

参考文献

Journal of the American Chemical Society, , vol. 136, # 11 p. 4287 - 4299

1112982-81-6+

73183-34-3联硼酸频那醇酯

1112983-23-9

参考文献

AMGEN INC.
Patent: WO2009/155121 A2, 2009 ;
Location in patent: Page/Page column 108-109 ;