1: With potassium acetate in 1,4-dioxane 0.25 h; 2: With (1,1'-bis(diphenylphosphino)ferrocene)palladium(II) dichloride in 1,4-dioxane; dichloromethane T=100°C; 2 h;
参考文献
AXYS PHARMACEUTICALS, INC.
Patent: WO2006/86609 A2, 2006 ;
Location in patent: Page/Page column 152-153 ;
WO 2006/086609 A2