联硼酸频那醇酯合成路线

参考文献

Chow, Wing Kin; So, Chau Ming; Lau, Chak Po; Kwong, Fuk Yee
Chemistry - A European Journal, 2011 , vol. 17, # 25 p. 6913 - 6917

5798-75-44-溴苯甲酸乙酯+

73183-34-3联硼酸频那醇酯

195062-62-54-(4,4,5,5-四甲基-1,3,2-二氧硼戊环-2-基)苯甲酸乙酯

参考文献

Gurung, Santosh K.; Kim, Soo Bae; Park, Haeil
Archives of Pharmacal Research, 2010 , vol. 33, # 12 p. 1919 - 1926

651780-02-85-溴-1H-吲唑-1-甲酸叔丁酯+

73183-34-3联硼酸频那醇酯

864771-44-85-(4,4,5,5-四甲基-1,3,2-二氧硼烷-2-基)-1H-吲哒唑-1-甲酸叔丁酯

参考文献

GLAXOSMITHKLINE LLC; CHAUDHARI, Amita, M.; HALLMAN, Jason; LAUDEMAN, Christopher, P.; MUSSO, David, Lee; PARRISH, Cynthia, A.
Patent: WO2011/66211 A1, 2011 ;
Location in patent: Page/Page column 69-70 ;
WO 2011/066211 A1

523-27-39,10-二溴蒽+

73183-34-3联硼酸频那醇酯

863992-56-79,10-蒽二硼酸二频哪酯

参考文献

Hiroki, Kazuaki; Kijima, Masashi
Chemistry Letters, 2005 , vol. 34, # 7 p. 942 - 943

887115-53-91-苯磺酰基-3- 碘 -1H- 吡咯[2,3-B]吡啶+

73183-34-3联硼酸频那醇酯

886547-94-01-苯磺酰基吡咯并吡啶-3-硼酸酯

参考文献

SMITHKLINE BEECHAM CORPORATION
Patent: WO2007/76423 A2, 2007 ;
Location in patent: Page/Page column 53 ;
WO 2007/076423 A2

880769-95-93-溴-1-甲基磺酰基-1H-吡咯并[2,3-B]吡啶+

73183-34-3联硼酸频那醇酯

886547-94-01-苯磺酰基吡咯并吡啶-3-硼酸酯

参考文献

Huang, Shenlin; Li, Ronghua; Connolly, Peter J.; Emanuel, Stuart; Middleton, Steven A.
Bioorganic and Medicinal Chemistry Letters, 2006 , vol. 16, # 18 p. 4818 - 4821

57883-25-73-溴-2-乙氧基吡啶+

73183-34-3联硼酸频那醇酯

848243-23-22-乙氧基吡啶-3-硼酸频哪醇酯

参考文献

PFIZER LIMITED; STORER, Robert, Ian; SWAIN, Nigel, Alan
Patent: WO2013/93688 A1, 2013 ;
Location in patent: Page/Page column 44-45 ;

630121-86-73-(三氟甲基磺酰氧基)-2H-吡咯-1(5h)-羧酸叔丁酯+

73183-34-3联硼酸频那醇酯

212127-83-83-(4,4,5,5-四甲基-1,3,2-二噁硼烷-2-基)-2,5-二氢-1H-吡咯-1-羧酸叔丁酯

参考文献

US2010/204265 A1, ;

Page/Page column 91; 92 ;

73183-34-3联硼酸频那醇酯+

188975-30-63,6-二氢-2H-吡喃-4-三氟甲烷磺酸盐