1: With potassium acetate in N,N-dimethyl-formamide 0.166667 h; 2: With dichloro(1,1'-bis(diphenylphosphanyl)ferrocene)palladium(II) dichloromethane adduct in N,N-dimethyl-formamide T=80°C;
potassium acetate; (1,1'-bis(diphenylphosphino)ferrocene)palladium(II) dichloride in N,N-dimethyl-formamide 0.333333 h; Microwave irradiation;
参考文献
THE GOVERNMENT OF THE UNITED STATES, as represented by the secretary of HEALTH AND HUMAN SERVICES
Patent: WO2007/124345 A2, 2007 ;
Location in patent: Page/Page column 25-26 ;