联硼酸频那醇酯合成路线

123-91-11,4-二氧六环

540752-87-23-[4-(叔丁氧基羰基)哌嗪-1-基]苯硼酸频那醇酯

参考文献

ASTRAZENECA AB
Patent: US2009/118305 A1, 2009 ;
US 20090118305 A1

540752-86-1+

73183-34-3联硼酸频那醇酯

540752-87-23-[4-(叔丁氧基羰基)哌嗪-1-基]苯硼酸频那醇酯

参考文献

Matasi, Julius J.; Caldwell, John P.; Zhang, Hongtao; Fawzi, Ahmad; Higgins, Guy A.; Cohen-Williams, Mary E.; Varty, Geoffrey B.; Tulshian, Deen B.
Bioorganic and Medicinal Chemistry Letters, 2005 , vol. 15, # 16 p. 3675 - 3678

73183-34-3联硼酸频那醇酯+

327030-39-74-(3-溴-苯基)-哌嗪-1-羧酸叔丁酯

540752-87-23-[4-(叔丁氧基羰基)哌嗪-1-基]苯硼酸频那醇酯

参考文献

Castillo, Marcos; Forns, Pilar; Erra, Montse; Mir, Marta; Lopez, Manel; Maldonado, Monica; Orellana, Adelina; Carreno, Cristina; Ramis, Isabel; Miralpeix, Montserrat; Vidal, Bernat
Bioorganic and Medicinal Chemistry Letters, 2012 , vol. 22, # 17 p. 5419 - 5423

53087-13-13-苄氧基溴苯+

73183-34-3联硼酸频那醇酯

765908-38-13-(苄氧基)苯硼酸频那醇酯

参考文献

The Procter and Gamble Company
Patent: US2007/209123 A1, 2007 ;
Location in patent: Page/Page column 8 ;

98-57-74-氯苯基甲基砜+

73183-34-3联硼酸频那醇酯

603143-27-74-(甲磺酰基)苯硼酸频哪醇酯

参考文献

Li, Pengbin; Fu, Chunling; Ma, Shengming
Organic and Biomolecular Chemistry, 2014 , vol. 12, # 22 p. 3604 - 3610

1007-15-43-溴-4-氟苯甲酮+

73183-34-3联硼酸频那醇酯

765916-70-9

参考文献

St. Jean Jr., David J.; Poon, Steve F.; Schwarzbach, Jamie L.
Organic Letters, 2007 , vol. 9, # 23 p. 4893 - 4896

849758-12-94-溴-3-氟苯甲酸甲酯+

73183-34-3联硼酸频那醇酯

603122-79-82-氟-4-(甲氧基羰基)苯硼酸频那醇酯

参考文献

Berthel, Steven Joseph; Chen, Li; Corbett, Wendy Lea; Feng, LiChun; Haynes, Nancy-Ellen; Kester, Robert Francis; So, Sung-Sau; Tilley, Jefferson Wright
Patent: US2011/144105 A1, 2011 ;
Location in patent: Page/Page column 70 ;

603122-83-4+

73183-34-3联硼酸频那醇酯

603122-79-82-氟-4-(甲氧基羰基)苯硼酸频那醇酯

参考文献

Imanishi, Masashi; Tomishima, Yasuyo; Itou, Shinji; Hamashima, Hitoshi; Nakajima, Yutaka; Washizuka, Kenichi; Sakurai, Minoru; Matsui, Shigeo; Imamura, Emiko; Ueshima, Koji; Yamamoto, Takao; Yamamoto, Nobuhiro; Ishikawa, Hirofumi; Nakano, Keiko; Unami, Naoko; Hamada, Kaori; Matsumura, Yasuhiro; Takamura, Fujiko; Hattori, Kouji
Journal of Medicinal Chemistry, 2008 , vol. 51, # 6 p. 1925 - 1944

62224-16-2+

73183-34-3联硼酸频那醇酯

709648-80-6

参考文献

MERCK SHARP and DOHME LIMITED; MERCK and CO., INC.
Patent: WO2007/85873 A1, 2007 ;
Location in patent: Page/Page column 18 ;
WO 2007/085873 A1

67237-53-0+

73183-34-3联硼酸频那醇酯

736987-75-0

参考文献

Zhao, Jie; Niu, Zhiqiang; Fu, Hua; Li, Yadong
Chemical Communications, 2014 , vol. 50, # 16 p. 2058 - 2060