联硼酸频那醇酯合成路线

参考文献

MERCK SHARP and DOHME CORP.; THOMPSON, Christopher, F.; SWEIS, Ramzi, F.
Patent: WO2011/28395 A1, 2011 ;
Location in patent: Page/Page column 20-21 ;

1270038-09-93-(4-甲氧基-3-(4,4,5,5-四甲基-1,3,2-二噁硼烷-2-基)苯基)丙酸甲酯

参考文献

MERCK SHARP and DOHME CORP.; LU, Zhijian; CHEN, Yi-Heng; SMITH, Cameron; LI, Hong; THOMPSON, Christopher, F.; SWEIS, Ramzi; SINCLAIR, Peter; KALLASHI, Florida; HUNT, Julianne; ADAMSON, Samantha, E.; DONG, Guizhen; ONDEYKA, Debra, L.; QIAN, Xiaoxia; SUN, Wanying; VACHAL, Petr; ZHAO, Kake
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Location in patent: Page/Page column 37; 38 ;
WO 2012/058187 A1

109-99-9四氢呋喃+

142-68-7四氢吡喃+

73183-34-3联硼酸频那醇酯

参考文献

Journal of the American Chemical Society, , vol. 134, # 30 p. 12422 - 12425

704-41-62-乙炔基-α,α,α-三氟甲苯+

73183-34-3联硼酸频那醇酯

1294009-25-82-三氟甲基-反式-beta-苯乙烯硼酸频那醇酯

参考文献

Zhao, Jie; Niu, Zhiqiang; Fu, Hua; Li, Yadong
Chemical Communications, 2014 , vol. 50, # 16 p. 2058 - 2060

704-41-62-乙炔基-α,α,α-三氟甲苯+

73183-34-3联硼酸频那醇酯

1294009-25-82-三氟甲基-反式-beta-苯乙烯硼酸频那醇酯

参考文献

Jang, Hwanjong; Zhugralin, Adil R.; Lee, Yunmi; Hoveyda, Amir H.
Journal of the American Chemical Society, 2011 , vol. 133, # 20 p. 7859 - 7871

30951-66-72-羟基-2-(3-溴苯基)丙烷+

73183-34-3联硼酸频那醇酯

1309980-11-72-(3-(4,4,5,5-四甲基-1,3,2-二噁硼烷-2-基)苯基)丙烷-2-醇

参考文献

SANOFI; ARNAUD, Joëlle; ARTIAGA, Martine; BARTH, Francis; HORTALA, Laurent; MARTINEZ, Serge; ROUX, Pascale
Patent: WO2013/87643 A1, 2013 ;
Location in patent: Page/Page column 15-16 ;

766-47-22-乙炔基甲苯+

73183-34-3联硼酸频那醇酯

1294009-26-92-甲基-beta-苯乙烯硼酸频那醇酯

参考文献

Jang, Hwanjong; Zhugralin, Adil R.; Lee, Yunmi; Hoveyda, Amir H.
Journal of the American Chemical Society, 2011 , vol. 133, # 20 p. 7859 - 7871

766-47-22-乙炔基甲苯+

73183-34-3联硼酸频那醇酯

1294009-26-92-甲基-beta-苯乙烯硼酸频那醇酯

参考文献

Jang, Hwanjong; Zhugralin, Adil R.; Lee, Yunmi; Hoveyda, Amir H.
Journal of the American Chemical Society, 2011 , vol. 133, # 20 p. 7859 - 7871

886374-01-22-甲氧基-3-氟-5-氯吡啶+

73183-34-3联硼酸频那醇酯

1310384-35-0

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AMGEN INC.; DRANSFIELD, Paul, John; GONZALEZ LOPEZ DE TURISO, Felix; KOHN, Todd, J.; PATTAROPONG, Vatee; SIMARD, Jillian, L.
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WO 2012/003283 A1

81971-39-35-溴-1-甲基-2(1H)-吡啶酮+

73183-34-3联硼酸频那醇酯

1002309-52-51-甲基-6-氧代-1,6-二氢吡啶-3-硼酸频那醇酯

参考文献

EP2168965 A1, ;

Page/Page column 33 ;
EP 2168965 A1