联硼酸频那醇酯合成路线

参考文献

BIOENERGENIX; MCCALL, John M.; ROMERO, Donna L.; KELLY, Robert C.
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Location in patent: Page/Page column 72 ;

452-73-32-氯-4-氟甲苯+

73183-34-3联硼酸频那醇酯

1126320-27-14-氯-2-氟-5-甲基苯硼酸频那醇酯

参考文献

Robbins, Daniel W.; Hartwig, John F.
Organic Letters, 2012 , vol. 14, # 16 p. 4266 - 4269

98-08-8三氟甲苯+

73183-34-3联硼酸频那醇酯

128796-39-44-三氟甲基苯硼酸+

1423-26-33-(三氟甲基)苯硼酸

参考文献

Yinghuai, Zhu; Yan, Koh Cheng; Jizhong, Luo; Hwei, Chong Siow; Hon, Yong Chun; Emi; Zhenshun, Su; Winata, Monalisa; Hosmane, Narayan S.; Maguire, John A.
Journal of Organometallic Chemistry, 2007 , vol. 692, # 20 p. 4244 - 4250

1183903-41-4+

73183-34-3联硼酸频那醇酯

1000801-76-21-(3-甲氧基丙基)-4-(4,4,5,5-四甲基-1,3,2-二噁硼烷-2-基)-1H-吡唑

参考文献

TAKEDA PHARMACEUTICAL COMPANY LIMITED; FENG, Jun; KEUNG, Walter; LARDY, Matthew
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WO 2010/129848 A2

1272756-07-64-(2-氯-4-溴苯基)吗啉+

73183-34-3联硼酸频那醇酯

1361110-63-53-氯-4-(4-吗啉基)苯硼酸频哪醇酯

参考文献

Trabanco, Andres A.; Tresadern, Gary; MacDonald, Gregor J.; Vega, Juan Antonio; De Lucas, Ana Isabel; Matesanz, Encarnacion; Garcia, Aranzazu; Linares, Maria Lourdes; Alonso De Diego, Sergio A.; Alonso, Jose Manuel; Oehlrich, Daniel; Ahnaou, Abdelah; Drinkenburg, Wilhelmus; MacKie, Claire; Andres, Jose Ignacio; Lavreysen, Hilde; Cid, Jose Maria
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25637-16-54-溴四氢吡喃+

73183-34-3联硼酸频那醇酯

1131912-76-9四氢吡喃-4-硼酸频哪醇酯

参考文献

Yi, Jun; Liu, Jin-Hui; Liang, Jun; Dai, Jian-Jun; Yang, Chu-Ting; Fu, Yao; Liu, Lei
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356560-80-06-溴-[1,2,4]三唑并[1,5-a]吡啶+

73183-34-3联硼酸频那醇酯

1160790-18-06-(4,4,5,5-四甲基-1,3,2-二噁硼烷-2-基)-[1,2,4]噻唑并[1,5-a]吡啶

参考文献

BAYER SCHERING PHARMA AKTIENGESELLSCHAFT; BAeRFACKER, Lars; KAST, Raimund; GRIEBENOW, Nils; MEIER, Heinrich; KOLKHOF, Peter; ALBRECHT-KUePPER, Barbara; NITSCHE, Adam; STASCH, Johannes-Peter; SCHNEIDER, Dirk; TEUSCH, Nicole; RUDOLPH, Joachim; WHELAN, James; BULLOCK, William; PLEASIC-WILLIAMS, Susan
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675109-26-96-溴异吲哚啉-1-酮+

73183-34-3联硼酸频那醇酯

1004294-80-71-异吲哚酮-6-硼酸频哪醇酯

参考文献

KUDOS PHARMACEUTICALS LIMITED
Patent: WO2008/23161 A1, 2008 ;
Location in patent: Page/Page column 117 ;
WO 2008/023161 A1

292638-85-8丙烯酸甲酯+

73183-34-3联硼酸频那醇酯

1150561-77-52-(甲氧基羰基)乙基硼酸频那醇酯

参考文献

LEK Pharmaceuticals d.d.; The designation of the inventor has not yet been filed
Patent: EP2647640 A1, 2013 ;
Location in patent: Paragraph 0072; 0073 ;

67-56-1甲醇+

292638-85-8丙烯酸甲酯+

73183-34-3联硼酸频那醇酯

1150561-77-52-(甲氧基羰基)乙基硼酸频那醇酯

参考文献

Knott, Kenneth; Fishovitz, Jennifer; Thorpe, Steven B.; Lee, Irene; Santos, Webster L.
Organic and Biomolecular Chemistry, 2010 , vol. 8, # 15 p. 3451 - 3456