联硼酸频那醇酯合成路线

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PFIZER LIMITED; ICAGEN, INC.; GREENER, Benjamin Scott; MARRON, Brian Edward; MILLAN, David Simon; RAWSON, David James; STORER, Robert Ian; SWAIN, Nigel Alan
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WO 2012/004714 A2

89402-43-75-氯-2,3-二氟吡啶+

73183-34-3联硼酸频那醇酯

1154579-82-42,3-二氟-5-(4,4,5,5-四甲基-1,3,2-二噁硼烷-2-基)吡啶

参考文献

EP2221301 A1, ;

Page/Page column 44 ;

851386-35-15-碘-2,3-二氟吡啶+

73183-34-3联硼酸频那醇酯

1154579-82-42,3-二氟-5-(4,4,5,5-四甲基-1,3,2-二噁硼烷-2-基)吡啶

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WO2013/74387 A1, ;

Page/Page column 43; 44 ;

110-87-23,4-二氢-2H-吡喃+

73183-34-3联硼酸频那醇酯

1046811-99-72-(3,4-二氢-2H-吡喃-5-基)-4,4,5,5-四甲基-1,3,2-二噁硼烷+

1025707-93-03,4-二氢-2H-吡喃-6-硼酸频那醇酯

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Miyaura, Norio
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1513-65-12,6-二氟吡啶+

73183-34-3联硼酸频那醇酯

1204333-58-32,6-二氟吡啶-4-硼酸频哪醇酯

参考文献

GLAXO GROUP LIMITED; ALDER, Catherine Mary; BALDWIN, Ian Robert; BARTON, Nicholas Paul; CAMPBELL, Amanda Jennifer; CHAMPIGNY, Aurelie Cecile; HARLING, John David; MAXWELL, Aoife Caitriona; SIMPSON, Juliet Kay; SMITH, Ian Edward David; TAME, Christopher John; WILSON, Caroline; WOOLVEN, James Michael
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WO 2011/110575 A1

73183-34-3联硼酸频那醇酯+

180695-79-8

1048970-17-7

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Yang, Chu-Ting; Zhang, Zhen-Qi; Tajuddin, Hazmi; Wu, Chen-Cheng; Liang, Jun; Liu, Jing-Hui; Fu, Yao; Czyzewska, Maria; Steel, Patrick G.; Marder, Todd B.; Liu, Lei
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884494-81-9+

73183-34-3联硼酸频那醇酯

1083168-95-9

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Burger, Matthew T.; Pecchi, Sabina; Wagman, Allan; Ni, Zhi-Jie; Knapp, Mark; Hendrickson, Thomas; Atallah, Gordana; Pfister, Keith; Zhang, Yanchen; Bartulis, Sarah; Frazier, Kelly; Ng, Simon; Smith, Aaron; Verhagen, Joelle; Haznedar, Joshua; Huh, Kay; Iwanowicz, Ed; Xin, Xiaohua; Menezes, Daniel; Merritt, Hanne; Lee, Isabelle; Wiesmann, Marion; Kaufman, Susan; Crawford, Kenneth; Chin, Michael; Bussiere, Dirksen; Shoemaker, Kevin; Zaror, Isabel; Maira, Sauveur-Michel; Voliva, Charles F.
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152684-30-5+

73183-34-3联硼酸频那醇酯

1083168-94-8

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WO2012/34526 A1, ;

Page/Page column 33 ;
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109-06-8+

73183-34-3联硼酸频那醇酯

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Obligacion, Jennifer V.; Semproni, Scott P.; Chirik, Paul J.
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