4-[6-[[5-溴-4-(环戊基氨基)-2-嘧啶]氨基]-3-吡啶]-1-哌嗪羧酸 1,1-二甲基乙酯合成路线 (共 1 条)
反应条件
1: in xylene; butan-1-ol
T=100 - 140°C;
2: With sodium hydroxide in water; ethyl acetate; xylene; butan-1-ol
参考文献
WARNER-LAMBERT COMPANY LLC
Patent: WO2004/65378 A1, 2004 ;
Location in patent: Page 31-32 ;
WO 2004/065378 A1