反应条件
1: KH poliamide resin, 4-(dimethylamino)pyridine, N-methylmorpholine, piperidine, 1percent TFA
2: 0.1 N HCl / tetrahydrofuran / 18 h / 25 °C
View Scheme
参考文献
Abraham; Nair; Kisliuk; Gaumont; Galivan
Journal of Medicinal Chemistry, 1990 , vol. 33, # 2 p. 711 - 717
