6-氯-N-(2-苯基乙基)嘧啶-4,5-二胺合成路线 (共 2 条)
反应条件
in formamide T=175°C; 4 h; Heating / reflux;
参考文献
Myriad Genetics, Incorporated
Patent: US2007/299258 A1, 2007 ;
Location in patent: Page/Page column 101 ;
反应条件
triethylamine in butan-1-ol
T=100°C; 12 h;
参考文献
Dang, Qun; Rydzewski, Robert M.; Cashion, Daniel K.; Erion, Mark D.
Tetrahedron Letters, 2008 , vol. 49, # 13 p. 2143 - 2145