4-溴苯乙胺合成路线

参考文献

Nguyen, Thanh Binh; Retailleau, Pascal; Al-Mourabit, Ali
Organic Letters, 2013 , vol. 15, # 20 p. 5238 - 5241

参考文献

Runyon, Scott P.; Mosier, Philip D.; Roth, Bryan L.; Glennon, Richard A.; Westkaemper, Richard B.
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73918-56-64-溴苯乙胺

181514-35-21-(7-溴-3,4-二氢异喹啉-2(1H)-基)-2,2,2-三氟乙酮

参考文献

Stokker
Tetrahedron Letters, 1996 , vol. 37, # 31 p. 5453 - 5456

50-00-0甲醛+

73918-56-64-溴苯乙胺+

407-25-0三氟乙酸酐

181514-35-21-(7-溴-3,4-二氢异喹啉-2(1H)-基)-2,2,2-三氟乙酮

参考文献

Pfizer Inc
Patent: US2005/182079 A1, 2005 ;
Location in patent: Page/Page column 11 ;

73918-56-64-溴苯乙胺+

407-25-0三氟乙酸酐

181514-21-6N-[2-(4-溴苯基)乙基]-2,2,2-三氟乙酰胺

参考文献

ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P ANGELETTI SPA
Patent: WO2004/87714 A1, 2004 ;
Location in patent: Page 71 ;
WO 2004/087714 A1

181514-21-6N-[2-(4-溴苯基)乙基]-2,2,2-三氟乙酰胺

参考文献

ASTRAZENECA AB
Patent: WO2004/60882 A1, 2004 ;
Location in patent: Page 35 ;
WO 2004/060882 A1

73918-56-64-溴苯乙胺+

79-30-1异丁酰氯

304664-15-1

参考文献

Bruncko, Milan; McClellan, William J.; Wendt, Michael D.; Sauer, Daryl R.; Geyer, Andrew; Dalton, Christopher R.; Kaminski, Michele A.; Weitzberg, Moshe; Gong, Jane; Dellaria, Joseph F.; Mantei, Robert; Zhao, Xumiao; Nienaber, Vicki L.; Stewart, Kent; Klinghofer, Vered; Bouska, Jennifer; Rockway, Todd W.; Giranda, Vincent L.
Bioorganic and Medicinal Chemistry Letters, 2005 , vol. 15, # 1 p. 93 - 98

50-00-0甲醛+

73918-56-64-溴苯乙胺+

407-25-0三氟乙酸酐

252331-63-86-溴-2-(三氟乙酰基)-1,2,3,4-四氢异喹啉

参考文献

Pfizer Inc
Patent: US2005/182079 A1, 2005 ;
Location in patent: Page/Page column 12 ;

73918-56-64-溴苯乙胺

891782-60-87-溴-3,4-二氢-2H-异喹啉-1-酮

参考文献

Kuduk, Scott D.; Chang, Ronald K.; Di Marco, Christina N.; Dipardo, Robert M.; Cook, Sean P.; Cato, Matthew J.; Jovanovska, Aneta; Urban, Mark O.; Leitl, Michael; Spencer, Robert H.; Kane, Stefanie A.; Hartman, George D.; Bilodeau, Mark T.
Bioorganic and Medicinal Chemistry Letters, 2011 , vol. 21, # 14 p. 4255 - 4258

5414-19-72,2'-二溴二乙醚+

73918-56-64-溴苯乙胺

736991-39-24-(4-溴苯乙基)吗啉

参考文献

Moss, Neil; Breitfelder, Steffen; Betageri, Raj; Cirillo, Pier F.; Fadra, Tazmeen; Hickey, Eugene R.; Kirrane, Thomas; Kroe, Rachel R.; Madwed, Jeffrey; Nelson, Richard M.; Pargellis, Christopher A.; Qian, Kevin C.; Regan, John; Swinamer, Alan; Torcellini, Carol
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