反应条件
1: 1H-indole-3-carboxylic acid With sodium hydride in DMF (N,N-dimethyl-formamide)
T=20°C; 0.166667 h;
2: 1-iodo-2,2-dimethylpropane in DMF (N,N-dimethyl-formamide)
T=80°C; 15 h;
参考文献
SANWA KAGAKU KENKYUSHO CO., LTD.
Patent: EP1595866 A1, 2005 ;
Location in patent: Page/Page column 19 ;