反应条件
1: 6-hydroxy-1,2,3,4-tetrahydro-2-quinolinone With 1,8-diazabicyclo[5.4.0]undec-7-ene in ethanol 6.5 h; Heating / refluxMolecular sieve; 2: 1-cyclohexyl-5-(4-chlorobutyl)-1,2,3,4-tetrazole in ethanol 6.5 h; Heating / reflux; Product distribution / selectivity;
参考文献
Naddaka, Vladimir; Davidi, Guy; Saeed, Shady; Arad, Oded; Kaspi, Joseph
Patent: US2005/222202 A1, 2005 ;
Location in patent: Page/Page column 5; 9 ;