2-氨基-2-(3-溴苯基)丙酸合成路线 (共 1 条)
反应条件
1: ammonia; ammonium chloride / methanol / 96 h / 20 °C
2: hydrogenchloride; water / 18 h / Reflux
View Scheme
参考文献
JANSSEN PHARMACEUTICA NV; TRABANCO-SUAREZ, Andres, Avelino; TRESADERN, Gary, John; MACDONALD, Gregor, James; VEGA RAMIRO, Juan, Antonio
Patent: WO2011/154374 A1, 2011 ;
WO 2011/154374 A1