1: With sodium hydroxide in tetrahydrofuran; water T=0°C; 0.5 h; 2: With acetic acid in tetrahydrofuran; water T=0°C; 3: With dihydrogen peroxide in tetrahydrofuran; water T=0 - 5°C;
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Song, Quanlai; Wang, Zhiwei; Sanghvi, Yogesh S.
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sodium cyanoborohydride in methanol Reductive amination;
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Lomenzo, Stacey A.; Izenwasser, Sari; Gerdes, Robert M.; Katz, Jonathan L.; Kopajtic, Theresa; Trudell, Mark L.
Bioorganic and Medicinal Chemistry Letters, 1999 , vol. 9, # 23 p. 3273 - 3276