C-(3,4-二氯-苯基)-c-苯基-甲基胺盐酸盐合成路线 (共 2 条)
反应条件
1: With acetic acid; zinc
T=20°C; 18 h;
2: With acetic acid in water
3: With hydrogenchloride; sodium carbonate
more than 3 stages;
参考文献
JANSSEN PHARMACEUTICA N.V.
Patent: WO2004/69809 A1, 2004 ;
Location in patent: Page 29 ;
WO 2004/069809 A1
反应条件
hydrogenchloride in isopropyl alcohol
参考文献
JANSSEN PHARMACEUTICA N.V.
Patent: WO2006/15986 A1, 2006 ;
Location in patent: Page/Page column 35-36 ;
WO 2006/015986 A1