1: benzenecarboximidamide hydrochloride With potassium hydroxide in dichloromethane; water 2: 1,2,3-triazine in 1,4-dioxane T=25°C; Diels-Alder reaction; 6 h; regioselective reaction;
参考文献
Anderson, Erin D.; Boger, Dale L.
Organic Letters, 2011 , vol. 13, # 9 p. 2492 - 2494
1: (1H)-pyrimidine With trifluoroacetic acid in dichloromethane; water 0.25 h; 2: 3,4,5-trimethoxyphenylboronic acid With iron sulphate heptahydrate; dipotassium peroxodisulfate in dichloromethane; water T=20°C; 5 h; 3: With sodium hydroxide in dichloromethane; water T=20°C; Overall yield = 65 percent;
参考文献
Bulletin of the Chemical Society of Japan, , vol. 87, # 2 p. 301 - 313
