反应条件
1: 200 mg / NaN3 / dimethylsulfoxide; H2O / 3 h / 90 °C 2: 1.) H2, 2.) HCl/Et2O / 1.) 10percent Pd/C / 1.) ethanol, 1 atm, r.t. View Scheme
参考文献
Kawamatsu; Asakawa; Saraie; Mizuno; Imamiya; Nishikawa; Hamuro
Arzneimittel-Forschung/Drug Research, 1980 , vol. 30, # 5 p. 751 - 758