2-(4-碘-1H-3-吡唑基)吡啶合成路线 (共 2 条)
反应条件
N-iodo-succinimide in DMF (N,N-dimethyl-formamide)
T=0 - 90°C;
参考文献
BIOGEN IDEC MA INC.
Patent: WO2004/72033 A2, 2004 ;
Location in patent: Page 35-36 ;
WO 2004/072033 A2
反应条件
triethylamine in chloroform
T=0°C; Heating / reflux;
参考文献
BIOGEN IDEC MA INC.
Patent: WO2004/72033 A2, 2004 ;
Location in patent: Page 36 ;
WO 2004/072033 A2