反应条件
1: 100 percent / thionyl chloride / 1.5 h / Heating
2: 79 percent / 5.5 h / Heating
3: 1.) NaOEt, 2.) HF 254-G silica gel / 1.) ethanol, 5 s, 2.) CH2Cl2
View Scheme
参考文献
Massy-Westropp, Ralph; Price, Martyn F.
Australian Journal of Chemistry, 1980 , vol. 33, # 2 p. 333 - 341