反应条件
1: 3-nitrobenzene-1,2-diol With sodium hydride in N,N,N',N',N'',N''-hexamethylphosphoric triamide
0.166667 h;
2: diiodomethane in N,N,N',N',N'',N''-hexamethylphosphoric triamide
0.5 h;
参考文献
CENTAURUS BIOPHARMA CO., LTD.; XIAO, Dengming; CHENG, Liang; LIU, Xijie; HU, Yuandong; XU, Xinhe; LIU, Zhihua; ZHANG, Lipeng; WU, Wei; WANG, Shulong; SHEN, Yu; LI, Gen; WANG, Yin; ZHAO, Sheng; LI, Chonglong; TANG, Jia; YU, Honghao
Patent: WO2012/92880 A1, 2012 ;
Location in patent: Page/Page column 61-62 ;
WO 2012/092880 A1