Givens, Richard S.; Matuszewski, Bogdan; Athey, Phillip S.; Robert Stoner
Journal of the American Chemical Society, 1990 , vol. 112, # 16 p. 6016 - 6021
Raju, P. V. K.; Adapa, Srinivas R.
Indian Journal of Chemistry, Section B: Organic Chemistry Including Medicinal Chemistry, 1992 , vol. 31, # 6 p. 363 - 365
4-(N,N-dimethlyamino)pyridine; dicyclohexyl-carbodiimide in dichloromethane
T=0 - 20°C; 4 h;
参考文献
Drewe, William C.; Nanjunda, Rupesh; Gunaratnam, Mekala; Beltran, Monica; Parkinson, Gary N.; Reszka, Anthony P.; Wilson, W. David; Neidle, Stephen
Journal of Medicinal Chemistry, 2008 , vol. 51, # 24 p. 7751 - 7767
1: With 4-(N,N-dimethlyamino)pyridine; dicyclohexyl-carbodiimide in dichloromethane; N,N-dimethyl-formamide
T=20°C; 15 h;
2: With 10 palladium on activated charcoal; hydrogen in methanol
T=20°C; 2 h;