反应条件
1: 94 percent / 4 M HCl / dioxane / 0.75 h 2: 1.) NH3, 2.) AcOH / 1.) CHCl3, 5 min, 2.) THF, 20 h 3: 60 percent / H2 / 5percent Pd/C / methanol; H2O / 24 h / 760 Torr View Scheme
参考文献
Mincev, Stoyan; Derdowska, Izabela; Kupryszewski, Gotfryd
Polish Journal of Chemistry, 1980 , vol. 54, # 3 p. 443 - 452