反应条件
1: 1.) PhLi / 1.) cyclohexane, Et2O, a) 0 deg C, 15 min, b) RT, 30 min, 1.) cyclohexane, Et2O, RT, 16 h 2: 89 percent / conc. HCl / tetrahydrofuran / a) 0 deg C, 20 min, b) RT, 3 h View Scheme
参考文献
Journal of Medicinal Chemistry, , vol. 42, # 4 p. 691 - 705