1: With lithium aluminium tetrahydride in tetrahydrofuran T=20°C; 48 h; Inert atmosphere; 2: With sodium hydroxide in tetrahydrofuran Inert atmosphere;
参考文献
ACADIA PHARMACEUTICALS, INC.; SCHLIENGER, Nathalie; THYGESEN, Mikkel; ULDAM, Henriette, Kold; SCHMELZER, Kara; TABATABAEI, Ali
Patent: WO2010/111353 A1, 2010 ;
Location in patent: Page/Page column 64-65 ;
WO 2010/111353 A1