反应条件
sodium hydride
1.) DMF, 1.5 h, 2.) DMF, 25 deg C, overnight; Yield given. Multistep reaction;
参考文献
Pelaprat, Didier; Oberlin, Robert; Le Guen, Irene; Roques, Bernard P.; Pecq, Jean-Bernard Le
Journal of Medicinal Chemistry, 1980 , vol. 23, # 12 p. 1330 - 1335