反应条件
1: 78 percent / dimethylformamide / 4 h / 80 °C
2: 1.) NaH, 2.) BuLi, 3.) Bf3*OEt2, 4.) KF
3: 90 percent / 10percent KOH / ethanol / 3 h / Heating
4: 81 percent / conc. HCl / methanol / 4 h / Heating
View Scheme
参考文献
Takeuchi, Naoki; Nakano, Takako; Goto, Kaori; Tobinaga, Seisho
Heterocycles, 1993 , vol. 35, # 1 p. 289 - 297