4-氟-3-(4,4,5,5-四甲基-1,3,2-二噁硼烷-2-基)苯甲酸甲酯合成路线 (共 1 条)
反应条件
potassium acetate; (1,1'-bis(diphenylphosphino)ferrocene)palladium(II) dichloride in dichloromethane; dimethyl sulfoxide
T=80°C; 2 h;
参考文献
VERTEX PHARMACEUTICALS INCORPORATED
Patent: WO2004/78733 A1, 2004 ;
Location in patent: Page 437 ;
WO 2004/078733 A1