1.1: piperidine / propan-2-ol / 3.5 h / 50 °C
1.2: 81 percent / NaOH / H2O; propan-2-ol / 4 h / 0 - 23 °C
2.1: 94 percent / trifluoroacetic anhydride / tetrahydrofuran; heptane / 23 - 55 °C
View Scheme
参考文献
Keen, Stephen P.; Cowden, Cameron J.; Bishop, Brian C.; Brands, Karel M. J.; Davies, Antony J.; Dolling, Ulf H.; Lieberman, David R.; Stewart, Gavin W.
Journal of Organic Chemistry, 2005 , vol. 70, # 5 p. 1771 - 1779