反应条件
1: diphenyl ether / 1 h / Heating
2: POCl3 / 1.17 h / 100 - 110 °C
3: a) 80-100 deg C, 1 h, b) 135-150 deg C, 8 h
View Scheme
参考文献
De, Dibyendu; Krogstad, Frances M.; Byers, Larry D.; Krogstad, Donald J.
Journal of Medicinal Chemistry, 1998 , vol. 41, # 25 p. 4918 - 4926