反应条件
1: indole; 2,2,2-trichloroacetyl chloride With pyridine in tetrahydrofuran T=0 - 20°C; 2: methanol With potassium hydroxide 6 h; Reflux;
参考文献
Lu, Wen-Jie; Switalska, Marta; Wang, Li; Yonezawa, Mizuki; El-Sayed, Ibrahim El-Tantawy; Wietrzyk, Joanna; Inokuchi, Tsutomu
Medicinal Chemistry Research, 2013 , vol. 22, # 9 p. 4492 - 4504