1: m-methoxypivanilide With n-butyllithium in tetrahydrofuran
T=0 - 22°C; 24 h;
2: oxirane in tetrahydrofuran
T=0°C;
参考文献
BOEHRINGER INGELHEIM INTERNATIONAL GMBH; BOEHRINGER INGELHEIM PHARMA GMBH and CO KG
Patent: WO2004/103996 A1, 2004 ;
Location in patent: Page 51-52 ;
WO 2004/103996 A1