反应条件
diphenylphosphoranyl azide; triethylamine in benzene
1.) 23 deg C, 30 min, 2.) reflux, 15 min;
参考文献
Reitz, Allen B.; Sonveaux, Etienne; Rosenkranz, Roberto P.; Verlander, Michael S.; Melmon, Kenneth L.; et al.
Journal of Medicinal Chemistry, 1985 , vol. 28, # 5 p. 634 - 642