3-[4-(三氟甲基)苯氧基]氮杂丁烷合成路线 (共 2 条)
反应条件
hydrogen; Pearlman's catalist in methanol T=60°C; P=2327.23 Torr; 18 h;
参考文献
Pfizer Inc.
Patent: US2010/190771 A1, 2010 ;
Location in patent: Page/Page column 28 ;
反应条件
di-isopropyl azodicarboxylate; triphenylphosphine in tetrahydrofuran T=20°C; 48 h;
参考文献
WO2012/76063 A1, ;
Page/Page column 60 ;
WO 2012/076063 A1