1-(3-氟苯基)-环丙胺合成路线 （共 2 条）
反应条件
1: With diphenyl phosphoryl azide; triethylamine in toluene
T=20°C; Curtius Rearrangement; 3 h; Heating / reflux;
2: With tert-butyl alcohol
20 h; Heating / reflux;
参考文献
BRISTOL-MYERS SQUIBB COMPANY
Patent: WO2004/43911 A2, 2004 ;
Location in patent: Page 49-50 ;
反应条件
hydrogenchloride in 1,4-dioxane; diethyl ether
T=20°C; 2 h;
参考文献
BRISTOL-MYERS SQUIBB COMPANY
Patent: WO2004/43911 A2, 2004 ;
Location in patent: Page 49; 51 ;
