反应条件
1: 4-bromophenylacetic acid With N-ethyl-N,N-diisopropylamine; HATU in N,N-dimethyl-formamide T=20°C; 0.25 h; 2: anhydrous cyclopropylamine in N,N-dimethyl-formamide T=20°C;
参考文献
Jones, Clifford D.; Andrews, David M.; Barker, Andrew J.; Blades, Kevin; Byth, Kate F.; Finlay, M. Raymond V.; Geh, Catherine; Green, Clive P.; Johannsen, Marie; Walker, Mike; Weir, Hazel M.
Bioorganic and Medicinal Chemistry Letters, 2008 , vol. 18, # 24 p. 6486 - 6489
