2,3-二氢-4-(4,4,5,5-四甲基-1,3,2-二氧硼烷)-1H-异吲哚-1-酮合成路线 （共 5 条）
反应条件
(1,1'-bis(diphenylphosphino)ferrocene)palladium(II) dichloride; potassium acetate in N,N-dimethyl-formamide T=80°C;
参考文献
Curtin, Michael L.; Frey, Robin R.; Heyman, H. Robin; Sarris, Kathy A.; Steinman, Douglas H.; Holmes, James H.; Bousquet, Peter F.; Cunha, George A.; Moskey, Maria D.; Ahmed, Asma A.; Pease, Lori J.; Glaser, Keith B.; Stewart, Kent D.; Davidsen, Steven K.; Michaelides, Michael R.
Bioorganic and Medicinal Chemistry Letters, 2004 , vol. 14, # 17 p. 4505 - 4509
反应条件
1: 94 percent / NBS; Bz2O2 / benzene 2: 87 percent / aq. NH3 / tetrahydrofuran 3: 63 percent / PdCl2(dppf); KOAc / dimethylformamide / 80 °C View Scheme
参考文献
Bioorganic and Medicinal Chemistry Letters, , vol. 14, # 17 p. 4505 - 4509
反应条件
1: Et3N 2: 94 percent / NBS; Bz2O2 / benzene 3: 87 percent / aq. NH3 / tetrahydrofuran 4: 63 percent / PdCl2(dppf); KOAc / dimethylformamide / 80 °C View Scheme
参考文献
Bioorganic and Medicinal Chemistry Letters, , vol. 14, # 17 p. 4505 - 4509
反应条件
1: SOCl2 2: Et3N 3: 94 percent / NBS; Bz2O2 / benzene 4: 87 percent / aq. NH3 / tetrahydrofuran 5: 63 percent / PdCl2(dppf); KOAc / dimethylformamide / 80 °C View Scheme
参考文献
Bioorganic and Medicinal Chemistry Letters, , vol. 14, # 17 p. 4505 - 4509
反应条件
1: 87 percent / aq. NH3 / tetrahydrofuran 2: 63 percent / PdCl2(dppf); KOAc / dimethylformamide / 80 °C View Scheme
参考文献
Bioorganic and Medicinal Chemistry Letters, , vol. 14, # 17 p. 4505 - 4509
