反应条件
1: 80 percent / Et3N / CH2Cl2 / 1 h / Ambient temperature
2: 97 percent / CuI, Pd(PPh3)4, n-PrNH2 / benzene / 3 h / Ambient temperature
View Scheme
参考文献
Okumura, Kunio; Shimazaki, Toshiyuki; Aoki, Yoji; Yamashita, Hiroyuki; Tanaka, Eishi; Banba, Shinichi; Yazawa, Kouhei; Kibayashi, Kenji; Banno, Hitoshi
Journal of Medicinal Chemistry, 1998 , vol. 41, # 21 p. 4036 - 4052