反应条件
1: N-(9-fluorenylmethoxycarbonyl)-L-aspartic acid-β-(tert-butyl)ester With 4-methyl-morpholine; N-methyl-N-(4,6-dimethoxy-2,4,6-triazin-2-yl)-morpholinium p-toluenosulphonate in acetonitrile T=0°C; 2 h; 2: 2,3,4,5,6-pentafluorophenol in acetonitrile T=0 - 20°C; 20 h;
参考文献
Politechnika Lodzka; Kaminski, Zbigniew; Kolesinska, Beata
Patent: EP1586566 A1, 2005 ;
Location in patent: Page/Page column 5-6 ;