N-(2,6-二甲基-4-氧代-1,4-二氢-5-嘧啶基)-4-甲基苯甲酰胺合成路线 (共 1 条)
反应条件
1: 1-Imino-ethanamine hydrochloride With sodium ethanolate in ethanol
T=20°C; 0.5 h;
2: 2-(4-methyl-benzoylamino)-3-oxo-butyric acid ethyl ester in ethanol
T=20°C; Further stages.;
参考文献
Norman; Chen; Fotsch; Hale; Han; Hurt; Jenkins; Kincaid; Liu; Lu; Moreno; Santora; Sonnenberg; Karbon
Journal of Medicinal Chemistry, 2000 , vol. 43, # 22 p. 4288 - 4312