5-氰基-2-氟苯硼酸频哪醇酯合成路线 (共 1 条)
反应条件
potassium acetate; (1,1'-bis(diphenylphosphino)ferrocene)palladium(II) dichloride in 1,4-dioxane T=100°C; Inert atmosphere;
参考文献
GLAXO GROUP LIMITED; BULLION, Ann, Marie; BUSCH-PETERSEN, Jakob; EVANS, Brian; NEIPP, Christopher, E.; MCCLELAND, Brent, W.; NEVINS, Neysa; WALL, Michael, D.
Patent: WO2011/25799 A1, 2011 ;
Location in patent: Page/Page column 50 ;
WO 2011/025799 A1