(1,1'-bis(diphenylphosphino)ferrocene)palladium(II) dichloride; potassium phosphate in 1,4-dioxane T=100°C; Suzuki coupling; 72 h;

(1,1'-bis(diphenylphosphino)ferrocene)palladium(II) dichloride; potassium phosphate in 1,4-dioxane T=100°C; Suzuki coupling; 72 h;

1: 6-(4,4,5,5-tetramethyl-[1,3,2]dioxaborolan-2-yl)-indole-1-carboxylic acid tert-butyl ester With diethylzinc in toluene T=70°C; 12 h; Inert atmosphere; 2: 3,4-dihydro-isoquinoline 2-oxide; diethylzinc With [(1S)-1-((S)-1-methylpropyl)-(2-morpholin-4-ylethyl)]carbamic acid tert-butyl ester in dichloromethane; toluene T=-30 - -20°C; 24.25 h; Inert atmosphere; 3: With methanol in dichloromethane; toluene T=-20°C; Inert atmosphere; optical yield given as percent eeenantioselective reaction;