1: With boron tribromide in hexane; dichloromethane
T=20°C; 1 h;
2: With ammonium chloride in hexane; dichloromethane
T=60°C; 1 h;
参考文献
Bernardo, Paul H.; Chai, Christina L. L.; Heath, Graham A.; Mahon, Peter J.; Smith, Geoffrey D.; Waring, Paul; Wilkes, Bronwyn A.
Journal of Medicinal Chemistry, 2004 , vol. 47, # 20 p. 4958 - 4963