反应条件
1: triethylamine / tetrahydrofuran / 0.33 h / 0 °C / Inert atmosphere
2: lithium azide / N,N-dimethyl-formamide / 8 h / 100 °C / Inert atmosphere
3: acetic acid / water / 20 °C / Inert atmosphere
View Scheme
参考文献
Sun, Jingbo; Liu, Xinyu; Li, Hongming; Duan, Ronghui; Wu, Jinchang
Helvetica Chimica Acta, 2012 , vol. 95, # 5 p. 772 - 779